- Indexed structures
- 3
- First release
- 6 Nov 2019
- Approved drugs
- 2
Written up here
Discovery of an Orally Bioavailable KRAS G12D Inhibitor_2
Casebook · 8 Mar 2026
2025 – Discovery of INCB159020, an Orally Bioavailable KRAS G12D Inhibitor
Casebook · 11 Aug 2025
All indexed structures
3 entries| Entry | Title | Method | Resolution | Released |
|---|---|---|---|---|
| 9E5D | Discovery of an Orally Biovailable KRAS G12D Inhibitor | X-ray | 1.36 Å | 22 Jan 2025 |
| 9E5F | Discovery of an Orally Bioavailable KRAS G12D Inhibitor | X-ray | 1.35 Å | 22 Jan 2025 |
| 6OIM | Crystal Structure of human KRAS G12C covalently bound to AMG 510 | X-ray | 1.65 Å | 6 Nov 2019 |